CORRECTION article

Front. Pharmacol., 04 May 2022

Sec. Pharmacology of Anti-Cancer Drugs

Volume 13 - 2022 | https://doi.org/10.3389/fphar.2022.907413

Corrigendum: Pharmacokinetics, Immunogenicity and Safety Study for SHR-1309 Injection and Perjeta® in Healthy Chinese Male Volunteers

    YC

    Yingzi Cui 1

    DC

    Dongyang Cui 2,3

    XR

    Xinran Ren 4,5

    XC

    Xuesong Chen 6

    GL

    Guangwen Liu 1

    ZL

    Zhengzhi Liu 1

    YW

    Yanli Wang 1

    XQ

    Xinyao Qu 1

    YZ

    Yicheng Zhao 5

    HY

    Haimiao Yang 1*

  • 1. Phase I Clinical Trial Laboratory, Affiliated Hospital of Changchun University of Chinese Medicine, Jilin, China

  • 2. Jiangsu Hengrui Medicine Co., Ltd., Lianyungang, China

  • 3. Shanghai Hengrui Pharmaceutical Co., Ltd., Shanghai, China

  • 4. School of Pharmacy, Jilin University, Jilin, China

  • 5. Clinical Medical College, Changchun University of Chinese Medicine, Jilin, China

  • 6. Jilin Province Honesty Medical Technology Consulting Co., Ltd., Jilin, China

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In the original article, there was a mistake in “Tables 2, 3” as published. “In Tables 2, 3, the AUC0-t and AUC0-∞ units were set to h*ng/ml by mistake.” The corrected “Tables 2, 3” appears below.

TABLE 2

SHR-1309 injection (N = 40)Perjeta® (N = 39)
Cmax (μg/ml)63.40 ± 15.1864.58 ± 17.17
AUC0-t (day*μg/mL)653.37 ± 133.65746.26 ± 197.06
AUC0-∞ (day*μg/mL)657.29 ± 133.29749.70 ± 198.23
Tmax (h)3.00 (0.99–48)1.50 (1–72)
t1/2z (day)7.29 ± 2.427.06 ± 2.11
Vss (mL/kg)70.92 ± 11.9166.04 ± 11.24
Vz (mL/kg)49.26 ± 16.8241.69 ± 10.94
CLz (mL/h/kg)0.20 ± 0.040.18 ± 0.04
λz (1/day)0.11 ± 0.030.11 ± 0.03
MRT0-t (day)14.78 ± 2.0815.61 ± 1.88
MRT0-∞ (day)15.12 ± 2.0115.87 ± 1.93
AUC%Extrap (%)0.64 ± 0.760.45 ± 0.46

The main PK parameters of SHR-1309 injection or Perjeta® after intravenous drip.

Mean ± SD was used to describe the parameters; Tmax was described by median (min max); Cmax, the maximum observed drug concentration in the plasma; AUC0-t, the AUC of the analyte in the plasma over the time interval from time zero to the last measurable concentration; AUC0-∞, the area under the curve from 0 to infinity; Tmax, the time from administration to the maximum observed concentration of the analyte in the plasma; t1/2z, the terminal half-life of the analyte in the plasma; Vss, the steady-state apparent distribution volume was measured after intravenous administration; Vz, distribution volume; CLz, clearance rate; λz, terminal rate constant in the plasma; MRT0-t, mean residence time from zero to the lowest detectable concentration; MRT0-∞, mean residence time extrapolated from zero to infinity; AUC%Extrap = [(AUC0-∞–AUC0-t)/AUC0-∞ × 100].

TABLE 3

PK parameterGeometric meanComparison
SHR-1309 injection (N = 40)Perjeta® (N = 39)Ratio%90% CI (%)
Cmax (μg/ml)61.9263.5397.4789.66–105.9
AUC0-t (day*μg/mL)639.65734.0787.1480.07–94.83
AUC0-∞ (day*μg/mL)643.88737.4387.3180.27–94.98
t1/2z (day)6.976.84101.8190.62–114.39
Vss (mL/kg)69.8364.47108.33101.19–115.96
Vz (mL/kg)46.8640.17116.67103.93–130.96
CLz (mL/h/kg)0.190.17114.59105.30–124.69
MRT0-t (day)14.6115.5893.7789.13–98.65
MRT0-∞ (day)14.6115.8494.5490.04–99.26

Results of the equivalence determination of the test drug and reference drug.

PK, pharmacokinetic; CI, confidence interval; Cmax, maximum observed drug concentration in the plasma; AUC0-t, the AUC of the analyte in the plasma over the time interval from time zero to the last measurable concentration; AUC0-∞, the area under the curve from 0 to infinity; t1/2z, the terminal half-life of the analyte in the plasma; Vss, steady-state apparent distribution volume was measured after intravenous administration; Vz, distribution volume; CLz, clearance rate; MRT0-t, mean residence time from zero to the lowest detectable concentration; MRT0-∞, mean residence time extrapolated from zero to infinity.

In the original article, there was an error. “The AUC0-t and AUC0-∞ units were set to h*ng/ml by mistake.”

A correction has been made to “Results,” “Pharmacokinetics,”:

“To evaluate the bioequivalence of SHR-1309 and Perjeta®, we performed PK analysis on two groups of subjects. The subjects were sampled at 21 time points before and after drug administration. Plasma drug concentration was detected by ELISA, and the data were fitted to form the average plasma drug concentration curve of SHR-1309 and Perjeta® (Figure 2A). The logarithmic transformation of the curve is shown in Figure 2B. At the same time, the plasma drug concentration of each subject in the two groups was fitted (Figures 2C,D). There was no significant difference in blood concentration between the two groups after administration. The primary evaluation parameters, secondary evaluation parameters and other pharmacokinetic parameters were obtained through calculation of plasma drug concentration (Table 2; Supplementary Table S1). The mean and standard deviation (SD) values of Cmax were 63.40 ± 15.18 μg/ml and 64.58 ± 17.17 μg/ml for SHR-1309 and Perjeta®, respectively, and the ratio of the geometric mean was 98.30%. The mean and SD values of AUC0-t were 653.37 ± 133.65 and 746.26 ± 197.06 day*μg/mL, respectively, and the ratio of the geometric mean was 88.41%. The mean and SD values of AUC0-∞ were 657.29 ± 133.29 and 749.70 ± 198.23 day*μg/mL, respectively, and the ratio of the geometric mean was 88.58%. Tmax was 1.50 and 3.00 h, respectively. The geometric mean values and ratios of all parameters are shown in Table 3. The primary pharmacokinetic parameters of SHR-1309 and Perjeta® were all up to the standard. Except for Vz, the 90% CI for all values fell within the 80%–125% range (Figure 3A). The PK parameter values of the two drugs were similar, and according to the PK evaluation standard of bioequivalence, SHR-1309 and Perjeta® are bioequivalent.”

The authors apologize for this error and state that this does not change the scientific conclusions of the article in any way. The original article has been updated.

Statements

Publisher’s note

All claims expressed in this article are solely those of the authors and do not necessarily represent those of their affiliated organizations, or those of the publisher, the editors and the reviewers. Any product that may be evaluated in this article, or claim that may be made by its manufacturer, is not guaranteed or endorsed by the publisher.

Summary

Keywords

perjeta®, pharmacokinetics, bioequivalence, immunogenicity, safety, SHR-1309 injection

Citation

Cui Y, Cui D, Ren X, Chen X, Liu G, Liu Z, Wang Y, Qu X, Zhao Y and Yang H (2022) Corrigendum: Pharmacokinetics, Immunogenicity and Safety Study for SHR-1309 Injection and Perjeta® in Healthy Chinese Male Volunteers. Front. Pharmacol. 13:907413. doi: 10.3389/fphar.2022.907413

Received

29 March 2022

Accepted

07 April 2022

Published

04 May 2022

Volume

13 - 2022

Edited and reviewed by

Wang Lingzhi, National University of Singapore, Singapore

Updates

Copyright

*Correspondence: Haimiao Yang,

†These authors have contributed equally to this work

This article was submitted to Pharmacology of Anti-Cancer Drugs, a section of the journal Frontiers in Pharmacology

Disclaimer

All claims expressed in this article are solely those of the authors and do not necessarily represent those of their affiliated organizations, or those of the publisher, the editors and the reviewers. Any product that may be evaluated in this article or claim that may be made by its manufacturer is not guaranteed or endorsed by the publisher.

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